1. |
(R)-Boc-β-Iodo-Ala-Ome |
93267-04-0 |
Eluxadoline |
4-Iodo-3,5-dimethyl benzonitrile |
1227311-09-2 |
2. |
Tert-butyl 3-(3-methylpyridin-2-yl)benzoate |
1083057-12-8 |
VX-809, Lumacaftor |
3-(6-Amino-3-methyl-pyridin-2-yl)-benzoic acid tert-butyl ester |
1083057-14-0 |
1-(2,2-Difluoro-benzo[1,3]dioxol-5-yl)-cyclopropane carboxylic acid |
862574-88-7 |
3. |
Benzofuran-6-carboxylic acid |
77095-51-3 |
Lifitegrast |
5,7-dichloro-2-BOC-1,2,3,4-tetrahydroisoquinoline-6-carboxylic acid |
851784-82-2 |
Methyl (S)-2-amino-3-(3-(methylsulfonyl)phenyl)propanoate hydrochloride |
851785-21-2 |
Benzyl (S)-2-amino-3-(3-(methylsulfonyl)phenyl)propanoate |
1194550-59-8 |
L-Phenylalanine, N-[(5,7-dichloro-1,2,3,4-tetrahydro-6-isoquinolinyl)carbonyl]-3-(methylsulfonyl)-phenylmethyl ester hydrochloride |
1194550-65-6 |
4. |
Ethyl 4-(2-chloropyrimidin-4-yl)benzoate |
499195-60-7 |
Momelotinib Dihydrochloride |
Ethyl 4-(2-(4-Morpholinophenylamino)pyrimidin-4-yl)benzoate |
1056634-62-8 |
Momelotinib |
1056634-68-4 |
5. |
Abemaciclib mesylate |
1231930-82-7 |
Abemaciclib |
5-((4-Ethylpiperazin-1-yl)methyl)pyridin-2-amine |
1180132-17-5 |
2-Bromopyridine-5-carbaldehyde |
149806-06-4 |
6-(2-chloro-5-fluoro-pyrimidin-4-yl)-4-fluoro-1-isopropyl-2-methyl-1H-benzo imidazole |
1231930-42-9 |
6-Bromo-4-fluoro-1-isopropyl-2-methyl-1H-benzo[d]imidazole |
1231930-33-8 |
6. |
N-Pyridin-2-yl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzamide |
1383385-64-5 |
Acalabrutinib, ACP-196 |
(2S)-2-(8-amino-1-bromoimidazo[1,5-a]pyrazin-3-yl)-1-Pyrrolidinecarboxylic acid phenylmethyl ester |
1420478-88-1 |
7. |
4-cyclopropylnaphthalen-1-amine hydrochloride |
1533519-92-4 |
RDEA 594, Lesinurad |
1-cyclopropyl-4-isothiocyanatonaphthalene |
878671-95-5 |
5-amino-4-(4-cyclopropyl-1-naphthalenyl)-2,4-dihydro-3H-1,2,4-Triazole-3-thione |
878671-96-6 |
4-(4-cyclopropylnaphthalen-1-yl)-1H-1,2,4-triazole-5(4H)-thione |
1533519-84-4 |
Methyl 2-[[4-(4-cyclopropylnaphthalen-1-yl)-4H-1,2,4-triazol-3-yl]thio]acetate |
1533519-85-5 |
8. |
2,4,5-Trifluorophenylacetic acid |
209995-38-0 |
Sitagliptin phosphate monohydrate |
Meldrum acid |
2033-24-1 |
3-(Trifluoromethyl)-5,6,7,8,-tetrahydro[1,2,4]triazolo[4,3-a]pyrazine HCl |
762240-92-6 |
9. |
3-Amino-1-adamantanol; 3-Amino-1-hydroxyadamantane |
702-82-9 |
Vildagliptin |
L-Prolinamide |
7531-52-4 |
(2S)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile |
207557-35-5 |
10. |
Tetrabenzyl voglibose |
115250-39-0 |
Voglibose |
11. |
N-Boc-4-oxo-L-proline |
84348-37-8 |
Teneligliptin Hydrobromide |
(2S)-4-oxo-2-(3-thiazolidinylcarbonyl)-1-pyrrolidinecarboxylic acid tert-butyl ester |
401564-36-1 |
1-(3-Methyl-1-phenyl-5-pyrazolyl)piperazine |
401566-79-8 |
12. |
(R)-3-BOC-Aminopiperidine |
309956-78-3 |
Linagliptin |
2-(chloro methyl)-4-methyl quinazoline |
109113-72-6 |
8-Bromo-7-(2-butynyl)-3,7-dihydro-3-methyl-1H-purine-2,6-dione |
666816-98-4 |
13. |
(R)-3-piperidinamine di-HCl |
334618-23-4 |
Alogliptin Benzoate |
6-Chloro-3-methyluracil |
4318-56-3 |
2-[(6-Chloro-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl)methyl]benzonitrile |
865758-96-9 |
14. |
Boc-3-Hydroxy-1-adamantyl-D-glycine |
361442-00-4 |
Saxagliptin HCl |
(1S,3S,5S)-3-(Aminocarbonyl)-2-azabicyclo[3.1.0]hexane-2-carboxylic acid tert-butyl ester |
361440-67-7 |
15. |
2,3,4,6-Tetrakis-O-trimethylsilyl-D-gluconolactone |
32384-65-9 |
Canagliflozin Hemihydrate |
16. |
2-(5-bromo-2-methylbenzyl)-5-(4-fluorophenyl)thiophene |
1030825-20-7 |
17. |
1-Cyclopropyl-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid ethyl ester |
112811-71-9 |
Moxifloxacin Hydrochloride |
18. |
(S,S)-2,8-diazabicyclo(4,3,0)nonane |
151213-42-2 |
19. |
4-Amino-5-imidazolecarboxamide hydrochloride |
72-40-2 |
Temozolomide |
20. |
2-Deoxy-D-Ribose |
553-67-5 |
Decitabine |
21. |
4,6-Dichloro-5-nitro-2-(propylthio)pyrimidine |
145783-14-8 |
Ticagrelor |
4,6-Dichloro-2-(PropylSulfanyl)-Pyrimidin-5-Amine |
145783-15-9 |
(1R,2S)-2-(3,4-Difluorophenyl)cyclopropanaminium (2R)-hydroxy(phenyl) ethanoate |
376608-71-8 |
(1R,2S)-2-(3,4-Difluorophenyl)-cyclopropan-1-amine HCl |
1156491-10-9 |
2-((3aR,4S,6R,6aS)-6-amino-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]dioxol-4- yloxy)ethanol L-tataric acid |
376608-65-0 |
22. |
4-octylphenethyl methane sulfonate |
162358-06-7 |
Fingolimod HCl |
1-(2-iodoethyl)-4-octylbenzene |
162358-07-8 |
Diethyl 2-acetamido-2-(4-octylphenethyl)malonate |
162358-08-9 |
N-(1-hydroxy-2-(hydroxymethyl)-4-(4-octylphenyl)butan-2-yl)acetamide |
249289-10-9 |
2-Acetoxymethyl-2-acetylamino-4-(4-octylphenyl)acetic acid butyl ester |
162358-09-0 |
Fingolimod Base |
162359-55-9 |
23. |
4-Cloromethyl-5-methyl-1,3-dioxol-2-one (DMDO-Cl) |
80841-78-7 |
Olmesartan Medoxomil |
24. |
Ethyl 4-(1-hydroxy-1-methylethyl)-2-propyl-imidazole-5-carboxylate |
144689-93-0 |
25. |
7-(4-Chlorobutoxy)-1H-quinolin-2-one |
913613-82-8 |
Brexpiprazole |
1-(Benzo[b]thiophen-4-yl)piperazine hydrochloride |
913614-18-3 |
1-(Benzo[b]thiophen-4-yl)piperazine |
846038-18-4 |
26. |
Methyl 2-bromomethyl-3-nitrobenzoate |
98475-07-1 |
Lenalidomide |
3-Aminopiperidine-2,6-dione hydrochloride (Pomalidomide intermediate as well) |
24666-56-6 |
27. |
4-(hydroxymethyl)-5-methyl-l,3-dioxol-2-one |
91526-18-0 |
Azilsartan |
1-(2-cyanobiphenyl-4-yl-methyl)- 2-ethoxybenzimidazole-7-carboxylic acid ethyl ester |
139481-44-0 |
28. |
R(+)-a-phenylethylamine, R(+)-a-methylbenzylamine |
3886-69-9 |
Pregabalin |
S-(-)-a-phenylethylamine, S(-)-a-methylbenzylamine |
2627-86-3 |
Glutaric anhydride |
108-55-4 |
3,4-Difluoronitrobenzene |
369-34-6 |
3,4-Difluoroaniline |
3863-11-4 |
5-Fluoro-2-oxindole |
56341-41-4 |
1-Iodo-4-nitrobenzene |
636-98-6 |
Diisopropyl azodicarboxylate (DIAD) |
2446-83-5 |
29. |
1-Methyl-Indozole-3-Carboxylic Acid / 1-MICA |
50890-83-0 |
Granisetron intermediates |
Endo-9-methyl-9-azabicyclo[3,3,1] -nonan-3 –amine / EMANA |
76272-56-5 |
Endo-9-methyl-9-azabicyclo[3,3,1] -nonan-3 -amine •2HCl / EMANA •2HCl |
135906-03-5 |
30. |
2-[(4-Chlorophenyl)acetyl]benzoic acid |
53242-76-5 |
Azelastine intermediates |
1-Methylhexahydroazepin-4-one hydrochloride |
19869-42-2 |
31. |
7-[2-(4-Fluoro-phenyl)-5-isopropyl-3-phenyl-4-(phenylcarbamoyl)pyrrol-1-yl]-3,5-dihydroxy-
heptanoic Acid tert-Butyl Ester / Atorvastatin tert-Butyl Ester |
134395-00-9 |
Atorvastatin intermediates |
(4R-Cis)-1,1-Dimethylethyl-6-[2-[2-(4-fluorophenyl)-5-(1-methylethyl)-3-phenyl-4-
[(phenylamino)carbonyl]-1H-pyrrol-1-yl]ethyl]-2,2-dimethyl-1,3-dioxane-4-acetate / L-1 |
125971-95-1 |
(4R-Cis)-1,1-dimethylethyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxane-4-acetate / Ats-8 |
125971-94-0 |
32. |
(+)-(3r, 5s), Tert-Butyl 7-[4-(4-Fluorophenyl)-6-Isopropyl-2-(N-Methyl-N-Methylsulphonylamino)-Pyrimidin-5-Yl]-3,5-Dihydroxy-6(E)-Heptenate / Rosuvastatin tert butyl ester |
355806-00-7 |
Rosuvastatin intermediates |
tert-Butyl (4R-cis)-6-[(acetyloxy)methyl]-2,2-dimethyl-1,3-dioxane-4-acetate / D5 |
154026-95-6 |
4-(4-Fluorophenyl)-6-isopropyl-2-[(N-methyl-n-methylsulfonyl)amino]pyrimidine-5-yl-methanol / Z-7 |
147118-36-3 |
33. |
5-(4-Chlorobutyl)-1-Cyclohexyl-1H-Tetrazole |
73963-42-5 |
Cilostazol intermediates |
3,4-dihydro-6-hydroxyquinolin-2(1H)-one |
54197-66-9 |
34. |
7,10-Dimethoxy-10-DAB III |
183133-94-0 |
Cabazitaxel intermediates |
35. |
4-Bromo-7-methoxy-1,3-benzodioxole-5-carboxylic acid methyl ester |
81474-46-6 |
Bifendate intermediates |
36. |
3-[(2R,5S)-5-(4-Fluorophenyl)-2-[(S)-[(4-fluorophenyl(amino)]][4-[trimethylsilyl]-
oxy]phenyl]methyl]-1-oxo-5-[(trimethylsily)-oxy]pentyl]-4-phenyl-(4S)-2-oxazolidinone / ZT-6 |
272778-12-8 |
Ezetimibe intermediates |
(3R,4S)-1-(4-Fluorophenyl)-3-[(3S)-3-(4-fluorophenyl)-3-hydroxypropyl]-4-[4-
(phenylmethoxy)phenyl]-2-azetidinone / E7 |
163222-32-0 |
37. |
(S)-1,2-diaminopropane dihydrochloride |
19777-66-3 |
Dexrazoxane intermediates |
38. |
3-(Trifluoromethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine hydrochloride |
762240-92-6 |
Sitagliptin intermediates |
Boc-(R)-3-Amino-4-(2,4,5-trifluorophenyl)butanoic acid |
486460-00-8 |
39. |
(S,S)-2,8 - Diazabicyclo (4,3,0) Nonane / Side chain |
151213-40-0 |
Moxifloxacin intermediates |
1-Cyclopropyl-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo-3 quinolinecarboxylic acid / Main chain |
112811-72-0 |
40. |
Methyl-2-(2,3-diclorobenzylidene)acetoacetate |
74073-22-6 |
Felodipine intermediates |
41. |
Phthaloyl Amlodipine |
88150-62-3 |
Amlodipine intermediates |
42. |
(3s,4r)-4-acetoxy-3-[(r)-1-(tert-butyldimethylsilyloxy)ethyl]azetidin-2-one / 4-AA |
76855-69-1 |
Carbapenem Basic KSM |
43. |
Diphenyl chlorophosphate / DPCP |
2524-64-3 |
44. |
2,2-Dimethyl-1,3-dioxane-4,6-dione / Meldrum's acid |
2033-24-1 |
45. |
p-Nitrobenzyl chloroformate |
4457-32-3 |
46. |
(2S,4S)-2-Dimethylaminocarboxyl-4-mercapto-1-p-nitrobenzyloxycarbonyl-pyrrolidine / 2S CIS |
[96034-64-9] |
Meropenem intermediates |
PNB(4R,5S,6S)-3-(Diphenyloxy)phosphoryloxy-6-[(1R)-1-hydroxyethyl]-4-methyl-7-oxo-1 azabicyclo[3,2,0]hept-2-ene-2-carboxylate / MAP |
[90776-59-3] |
47. |
1-Naphthyl acetonitrile |
132-75-2 |
Naphazoline intermediates |
48. |
N-[1-(S)-(Ethoxycarbonyl)-3-phenylpropyl]-L-alanine |
82717-96-2 |
Enalapril intermediates |
49. |
2-(1-(ethylsulfonyl)azetidin-3-ylidene)acetonitrile |
1187595-85-2 |
Baricitinib intermediates |
tert-Butyl 3-(cyanomethylene)azetidine-1-carboxylate |
1153949-11-1 |
1-Boc-pyrazole-4-boronic acid pinacol ester |
552846-17-0 |
Ethanesulfonyl Chloride |
594-44-5 |
50. |
7-Phenyl acetamido-3-Hydroxy-3-Cephem-4-Carboxylic acid Diphenylmethyl ester / GHYH |
54639-48-4 |
Ceftizoxime intermediates |
7-Amino-3-nor-3-cephem-4-carboxylic acid / 7-ANCA |
36923-17-8 |
51. |
5-Mercapto-1H-tetrazole-1-acetic acid / MTAA |
57658-36-3
|
Ceforanide intermediates |
2-Aminnomethyl phenyl acetic acid/AMPAA |
40851-65-8
|
52. |
2-Mercapto-5-methyl-1,3,4-thiadiazole / MMTD |
29490-19-5 |
Cefazolin intermediates |
1H-Tetrazol yl-1-acetic aid /TAA |
21732-17-2 |
53. |
(Z)-2-(5-Amino-1,2,4-Thiadiazol-3-yl)-2-Ethoxyiminoacetic Acid / ATDE |
75028-24-9 |
Ceftaroline intermediates |
4-(4-Pyridyl)thiazole-2-thiol / PTT |
77168-63-9 |
54. |
Boron Trifluoride Acetonitrile Complex |
420-16-6 |
Fine chemicals |
Boron Trifluoride DiMethyl Phthalate Complex |
N/A |
Boron Trifluoride |
7637-07-2 |